Efficient oxidation of cysteine and glutathione catalyzed by a dinuclear areneruthenium trithiolato anticancer complex.

نویسندگان

  • Federico Giannini
  • Georg Süss-Fink
  • Julien Furrer
چکیده

The highly cytotoxic diruthenium complex [(p-MeC(6)H(4)Pr(i))(2)Ru(2)(SC(6)H(4)-p-Me)(3)](+) (1), water-soluble as the chloride salt, is shown to efficiently catalyze oxidation of the thiols cysteine and glutathione to give the corresponding disulfides, which may explain its high in vitro anticancer activity.

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عنوان ژورنال:
  • Inorganic chemistry

دوره 50 21  شماره 

صفحات  -

تاریخ انتشار 2011